4
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12320 | ORL1 antagonist 1 | Opioid Receptor | |
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM). | |||
T6553 | JTC-801 | JTC 801,JTC801 | Opioid Receptor |
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ. | |||
T21999 | (±)-J 113397 | ||
(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM). J-113397 inhibited nociceptin/orphanin FQ-stimulated GTPγS binding to CHO cells expressing ORL1 with an IC 50... | |||
T75907 | Ac-RYYRIK-NH2 TFA | ||
Ac-RYYRIK-NH2 TFA acts as both a potent partial agonist for ORL1 when transfected in CHO cells (K d = 1.5 nM) and an endogenous ligand of ORL1. Moreover, it serves as a specific antagonist that inhibits G protein activat... |