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Search Results for " orl1 antagonist 1 "

4

Compounds

Cat No. Product Name Synonyms Targets
T12320 ORL1 antagonist 1 Opioid Receptor
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
T6553 JTC-801 JTC 801,JTC801 Opioid Receptor
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.
T21999 (±)-J 113397
(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM). J-113397 inhibited nociceptin/orphanin FQ-stimulated GTPγS binding to CHO cells expressing ORL1 with an IC 50...
T75907 Ac-RYYRIK-NH2 TFA
Ac-RYYRIK-NH2 TFA acts as both a potent partial agonist for ORL1 when transfected in CHO cells (K d = 1.5 nM) and an endogenous ligand of ORL1. Moreover, it serves as a specific antagonist that inhibits G protein activat...
TargetMol